GM 1489 N-[(2R)-2-(Carboxymethyl)-4-methylpentanoyl]-L-tryptophan-(S)-methyl-benzylamide This product has been discontinued. A potent broad-range inhibitor of matrix metalloproteinases (MMPs). Inhibits MMPs in vitro (Ki = 0.2 nM for MMP-1; Ki = 500 nM for MMP-2; Ki = 20 µM for MMP-3; Ki = 100 nM for MMP-8; and Ki = 100 nM for MMP-9). Also reduces the inflammatory and the hyperproliferative responses that occur following topical phorbol ester application. 产品信息 Form Off-white solid Primary Target MMP-1 Primary Target Ki 0.2 nM Secondary target Ki = 500 nM for MMP-2; Ki = 20 µM for MMP-3; Ki = 100 nM for MMP-8; and Ki = 100 nM for MMP-9 Molar mass 463.6 Purity ≥95% by HPLC Solubility DMSO Chemical formula C27H33N3O4 CAS number 170905-75-6 商店和运输信息 Storage -20°C Ship Ambient Temperature Only Standard Handling
