InSolution Casein Kinase II Inhibitor III, TBCA

InSolution™ Casein Kinase II Inhibitor III, TBCA
A cell-permeable tetrabrominated cinnamic acid compound that acts as a potent and ATP-competitive inhibitor of Casein Kinase II (IC50 = 110 nM, Ki = 77 nM) with greater selectivity than TBB (Cat. No. 218697 and Cat. No. 218708) and DMAT (Cat. No. 218699 and Cat. No. 218706) against a panel of 28 commonly studied kinases. Shown to efficiently induce apoptosis in Jurkat cells (DC50 = 7.7 µM). The solid form of this compound (Cat. No. 218710) is also available.
产品信息
Form  Liquid
Formulation  A 25 mM (5 mg/431 µL) solution of Casein Kinase II Inhibitor III, TBCA (Cat. No. 218710) in DMSO.
Primary Target  CKII
Molar mass  463.8
Protect from Light  是的
Hygrocopic  是的
Avoid freeze/thaw  是的
Packaged under inert gas  是的
Cell permeable  是的
Reversible  是的
Purity  ≥90% by HPLC
CAS number  934358-00-6
商店和运输信息
Storage  ≤ -70°C
Ship  Dry Ice Only
Irritant
安全标示
S Phrase  S: 26-36
In case of contact with eyes, rinse immediately with plenty of water and seek medical advice.
Wear suitable protective clothing.
R Phrase  R: 36/38
Irritating to eyes and skin.