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Bikinin
A highly specific inhibitor for the 7 Arabidopsis GSK-3 like kinase
Product Overview
Product Name: Bikinin
Alternate Name/Synonyms: 4-((5-Bromo-2-pyridinyl)amino)-4-oxobutanoic acid; Arabidopsis GSK-3 Inhibitor
Description: Cell-permeable. A highly specific inhibitor for the 7 Arabidopsis GSK-3 like kinase that activates brassinosteroid (BR) signaling downstream of the BR receptor. Bikinin directly binds the GSK3 BIN2 and acts as an ATP-competitive inhibitor. Furthermore, bikinin inhibits the activity of six other Arabidopsis GSK3s.
Peptide Sequence: N/A
Appearance: White solid
Formulation: N/A
CAS Number: 188011-69-0
Molecular Formula: C₉H₉BrN₂O₃
Molecular Weight: 273.08
Purity: ≥95% by HPLC
Solubility:DMSO ( 5 mg/ml)
Storage Temp.: -20°C
Shipping Conditions: gel pack
Handling: Protect from air and light
SMILES: C1=CC(=NC=C1Br)NC(=O)CCC(=O)O
InChi: InChI=1S/C9H9BrN2O3/c10-6-1-2-7(11-5-6)12-8(13)3-4-9(14)15/h1-2,5H,3-4H2,(H,14,15)(H,11,12,13)
InChi Key: XFYYQDHEDOXWGA-UHFFFAOYSA-N
PubChem CID: 647833
MDL Number: MFCD00116442
USAGE: For Research Use Only! Not For Use in Humans. |