M.Wt:412.01Formula:C20H25NO2S2.HClSolubility:Soluble to 50 mM in water and to 100 mM in DMSOPurity:>99 %Storage:Desiccate at RTCAS No:[145821-59-6]Biological ActivityGABA uptake inhibitor (IC50 = 67 nM in vivo). Exhibits high affinity and selectivity for the GAT-1 GABA transporter. Anticonvulsant; also attenuates established dynorphin-induced allodynia in a mouse model after systemic administration. Chemical Name: (3R)-1-[4,4-Bis(3-methyl-2-thienyl)-3-butenyl]-3-piperidinecarboxylic acid hydrochloride
