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产品信息
CAS number 1258003-96-1
Storage -20°C
A potent, reversible inhibitor of granzyme B and caspase-8 (Ki = 1 nM). Also inhibits caspase-1 (<6 nM), caspase-6 (5.6 nM), and caspase-10 (27 nM).
Peptide Sequence Ac-Ile-Glu-Thr-Asp-CHO
Form White lyophilized solid
Primary Target caspase-8
Primary Target Ki 1 nM
Secondary target caspase-1 (<6 nM), caspase-6 (5.6 nM), and caspase-10 (27 nM)
Reversible 是的
Purity ≥95% by HPLC
Chemical formula C21H34N4O10 |